Kerim Babaoglu : rechercher sur Z-Library

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1

Validation of Molecular Docking Programs for Virtual Screening against Dihydropteroate Synthase

Hevener, Kirk E., Zhao, Wei, Ball, David M., Babaoglu, Kerim, Qi, Jianjun, White, Stephen W., Lee, Richard E.

Journal:

Journal of Chemical Information and Modeling

Année:

2009

Langue:

english

Fichier:

PDF, 4.13 MB

english, 2009

2

Novel Inhibitors of an Emerging Target in Mycobacterium tuberculosis; Substituted Thiazolidinones as Inhibitors of dTDP-Rhamnose Synthesis.

Kerim Babaoglu, Mark A. Page, Victoria C. Jones, Michael R. McNeil, Changjiang Dong, James H. Naismith, Richard E. Lee

Journal:

Année:

2003

Fichier:

PDF, 85 KB

2003

3

Novel inhibitors of an emerging target in Mycobacterium tuberculosis; substituted thiazolidinones as inhibitors of dTDP-rhamnose synthesis

Kerim Babaoglu, Mark A. Page, Victoria C. Jones, Michael R. McNeil, Changjiang Dong, James H. Naismith, Richard E. Lee

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2003

Langue:

english

Fichier:

PDF, 228 KB

english, 2003

4

Deconstructing fragment-based inhibitor discovery

Babaoglu, Kerim, Shoichet, Brian K

Journal:

Nature Chemical Biology

Année:

2006

Langue:

english

Fichier:

PDF, 289 KB

english, 2006

5

Crystal Structure of 7,8-Dihydropteroate Synthase from Bacillus anthracis: Mechanism and Novel Inhibitor Design

Kerim Babaoglu, Jianjun Qi, Richard E. Lee, Stephen W. White

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 667 KB

english, 2004

6

Mutation of a Conserved Active Site Residue Converts Tyrosyl-DNA Phosphodiesterase I into a DNA Topoisomerase I-dependent Poison

Xiaoping He, Robert C.A.M. van Waardenburg, Kerim Babaoglu, Allen C. Price, Karin C. Nitiss, John L. Nitiss, Mary-Ann Bjornsti, Stephen W. White

Journal:

Journal of Molecular Biology

Année:

2007

Langue:

english

Fichier:

PDF, 1.29 MB

english, 2007

7

Design, Synthesis, Crystal Structures, and Antimicrobial Activity of Sulfonamide Boronic Acids as β-Lactamase Inhibitors

Eidam, Oliv, Romagnoli, Chiara, Caselli, Emilia, Babaoglu, Kerim, Pohlhaus, Denise Teotico, Karpiak, Joel, Bonnet, Richard, Shoichet, Brian K., Prati, Fabio

Journal:

Journal of Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 3.19 MB

english, 2010

8

O -Aryloxycarbonyl Hydroxamates: New β-Lactamase Inhibitors That Cross-Link the Active Site

Wyrembak, Pauline N., Babaoglu, Kerim, Pelto, Ryan B., Shoichet, Brian K., Pratt, R. F.

Journal:

Journal of the American Chemical Society

Année:

2007

Langue:

english

Fichier:

PDF, 122 KB

english, 2007

9

A High-Throughput Screen for Aggregation-Based Inhibition in a Large Compound Library

Feng, Brian Y., Simeonov, Anton, Jadhav, Ajit, Babaoglu, Kerim, Inglese, James, Shoichet, Brian K., Austin, Christopher P.

Journal:

Journal of Medicinal Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 252 KB

english, 2007

10

Comprehensive Mechanistic Analysis of Hits from High-Throughput and Docking Screens against β-Lactamase

Babaoglu, Kerim, Simeonov, Anton, Irwin, John J., Nelson, Michael E., Feng, Brian, Thomas, Craig J., Cancian, Laura, Costi, M. Paola, Maltby, David A., Jadhav, Ajit, Inglese, James, Austin, Christophe

Journal:

Journal of Medicinal Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 1.42 MB

english, 2008

11

Structural Studies of Pterin-Based Inhibitors of Dihydropteroate Synthase

Hevener, Kirk E., Yun, Mi-Kyung, Qi, Jianjun, Kerr, Iain D., Babaoglu, Kerim, Hurdle, Julian G., Balakrishna, Kanya, White, Stephen W., Lee, Richard E.

Journal:

Journal of Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 4.40 MB

english, 2010

12

Structure and ligand-binding mechanism of the human OX1 and OX2 orexin receptors

Yin, Jie, Babaoglu, Kerim, Brautigam, Chad A, Clark, Lindsay, Shao, Zhenhua, Scheuermann, Thomas H, Harrell, Charles M, Gotter, Anthony L, Roecker, Anthony J, Winrow, Christopher J, Renger, John J, Co

Journal:

Nature Structural and Molecular Biology

Année:

2016

Langue:

english

Fichier:

PDF, 2.09 MB

english, 2016

13

The HIV-1 Reverse Transcriptase M184I Mutation Enhances the E138K-Associated Resistance to Rilpivirine and Decreases Viral Fitness

Kulkarni, Rima, Babaoglu, Kerim, Lansdon, Eric B., Rimsky, Laurence, Van Eygen, Veerle, Picchio, Gaston, Svarovskaia, Evguenia, Miller, Michael D., White, Kirsten L.

Journal:

JAIDS Journal of Acquired Immune Deficiency Syndromes

Année:

2012

Langue:

english

Fichier:

PDF, 311 KB

english, 2012

14

Investigation of orexin-2 selective receptor antagonists: Structural modifications resulting in dual orexin receptor antagonists

Skudlarek, Jason W., DiMarco, Christina N., Babaoglu, Kerim, Roecker, Anthony J., Bruno, Joseph G., Pausch, Mark A., O'Brien, Julie A., Cabalu, Tamara D., Stevens, Joanne, Brunner, Joseph, Tannenbaum,

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2017

Langue:

english

Fichier:

PDF, 1.04 MB

english, 2017

15

Examining the Feasibility of Using Free Energy Perturbation (FEP+) in Predicting Protein Stability

Ford, Melissa Coates, Babaoglu, Kerim

Journal:

Journal of Chemical Information and Modeling

Année:

2017

Langue:

english

Fichier:

PDF, 1.46 MB

english, 2017

16

Structure-guided discovery of a novel, potent, and orally bioavailable 3,5-dimethylisoxazole aryl-benzimidazole BET bromodomain inhibitor

Sperandio, David, Aktoudianakis, Vangelis, Babaoglu, Kerim, Chen, Xiaowu, Elbel, Kristyna, Chin, Gregory, Corkey, Britton, Du, Jinfa, Jiang, Bob, Kobayashi, Tetsuya, Mackman, Richard, Martinez, Ruben,

Journal:

Bioorganic & Medicinal Chemistry

Année:

2018

Langue:

english

Fichier:

PDF, 1.26 MB

english, 2018

17

Characterization of potent RSV neutralizing antibodies isolated from human memory B cells and identification of diverse RSV/hMPV cross-neutralizing epitopes

Xiao, Xiao, Tang, Aimin, Cox, Kara S., Wen, Zhiyun, Callahan, Cheryl, Sullivan, Nicole L., Nahas, Deborah D., Cosmi, Scott, Galli, Jennifer D., Minnier, Michael, Verma, Deeptak, Babaoglu, Kerim, Su, H

Journal:

Année:

2019

Langue:

english

Fichier:

PDF, 5.74 MB

english, 2019